Tag «KRP 114V»

Vibegron ビベグロン

It’s only fair to share…   Vibegron, MK-4618, KRP 114V UNII-M5TSE03W5U; M5TSE03W5U; D10433 1190389-15-1;  cas no Molecular Formula: C26H28N4O3   Molecular Weight: 444.52552 Merck Sharp & Dohme Corp.  INNOVATOR phase 2 for the treatment of overactive bladder  (6S)-N-[4-([(2S,5R)-5-[(R)-Hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl)phenyl]-4-oxo-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide (6S)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-4-oxo-7,8-dihydro-6H-pyrrolo[1,2-a]pyrimidine-6-carboxamide Target-based Actions Beta 3 adrenoceptor agonist Indications Overactive bladder; Urinary incontinence UPDATE 2018/9/21  pmda Beova JAPAN 2018Kyorin Pharmaceutical, under license …