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IMIPRIDONE

It’s only fair to share… IMIPRIDONE CAS No. : 1616632-77-9 Molecular Weight, 386.4964 Related CAS #: 41276-02-2 (TIC10 isomer)   1616632-77-9 (free base)   1638178-82-1 (HCl)   1777785-71-3 (HBr)   2007141-57-1 (2HBr) TIC 10, 0NC 201, OP 10 Synonym: ONC201; ONC 201; ONC-201; NSC350625; NSC-350625; NSC 350625; TIC10; TIC 10; TIC-10; TRAIL inducing compound 10; imipridone 7-benzyl-4-(2-methylbenzyl)-1,2,6,7,8,9-hexahydroimidazo[1,2-a]pyrido[3,4-e]pyrimidin-5(4H)-one 2,4,6,7,8,9-Hexahydro-4-((2-methylphenyl)methyl)-7-phenylmethyl)imidazo)(1,2-a)pyrido(3,4-e)pyrimidin-5(1H)-one ONC-201 Dihydrochloride C24H28Cl2N4O 459.4 UNII-53VG71J90J …

Tirzepatide

It’s only fair to share… YXEGTFTSDY SIXLDKIAQK AFVQWLIAGG PSSGAPPPS Tirzepatide チルゼパチド LY3298176, Formula C225H348N48O68 CAS 2023788-19-2 Mol weight 4813.4514 FDA APPROVED 2022/5/13, Mounjaro Class Antidiabetic agent GLP-1 receptor agonist Efficacy Antidiabetic, Gastric inhibitory polypeptide receptor agonist, Glucagon-like peptide 1 (GLP-1) receptor agonist   Disease Type 2 diabetes mellitus L-Serinamide, L-tyrosyl-2-methylalanyl-L-α-glutamylglycyl-L-threonyl-L-phenylalanyl-L-threonyl-L-seryl-L-α-aspartyl-L-tyrosyl-L-seryl-L-isoleucyl-2-methylalanyl-L-leucyl-L-α-aspartyl-L-lysyl-L-isoleucyl-L-alanyl-L-glutaminyl-N6-[(22S)-22,42-dicarboxy-1,10,19,24-tetraoxo-3,6,12,15-tetraoxa-9,18,23-triazadotetracont-1-yl]-L-lysyl-L-alanyl-L-phenylalanyl-L-valyl-L-glutaminyl-L-tryptophyl-L-leucyl-L-isoleucyl-L-alanylglycylglycyl-L-prolyl-L-seryl-L-serylglycyl-L-alanyl-L-prolyl-L-prolyl-L-prolyl- Other Names L-Tyrosyl-2-methylalanyl-L-α-glutamylglycyl-L-threonyl-L-phenylalanyl-L-threonyl-L-seryl-L-α-aspartyl-L-tyrosyl-L-seryl-L-isoleucyl-2-methylalanyl-L-leucyl-L-α-aspartyl-L-lysyl-L-isoleucyl-L-alanyl-L-glutaminyl-N6-[(22S)-22,42-dicarboxy-1,10,19,24-tetraoxo-3,6,12,15-tetraoxa-9,18,23-triazadotetracont-1-yl]-L-lysyl-L-alanyl-L-phenylalanyl-L-valyl-L-glutaminyl-L-tryptophyl-L-leucyl-L-isoleucyl-L-alanylglycylglycyl-L-prolyl-L-seryl-L-serylglycyl-L-alanyl-L-prolyl-L-prolyl-L-prolyl-L-serinamide Tirzepatide is an agonist of human …

CLOSANTEL

It’s only fair to share… CLOSANTEL Closantel 57808-65-8 N-(5-chloro-4-((4-chlorophenyl)(cyano)methyl)-2-methylphenyl)-2-hydroxy-3,5-diiodobenzamide MW 663.1, C22H14Cl2I2N2O2   Closantel Sodium CAS NO. 61438-64-0 FORMULA C22H13Cl2I2N2O2.Na M. WT 685.06 Closantel CAS Registry Number: 57808-65-8 CAS Name: N-[5-Chloro-4-[(4-chlorophenyl)cyanomethyl]-2-methylphenyl]-2-hydroxy-3,5-diiodobenzamide Manufacturers’ Codes: R-31520 Trademarks: Flukiver (Janssen); Seponver (Ethnor) Molecular Formula: C22H14Cl2I2N2O2, Molecular Weight: 663.07 Percent Composition: C 39.85%, H 2.13%, Cl 10.69%, I 38.28%, N 4.22%, O 4.83% Literature References: Salicylanilide derivative. Prepn: M. …

MONENSIN

It’s only fair to share… モネンシン; MONENSIN Elancoban [veterinary] (TN) Molecular FormulaC36H62O11 Average mass670.871 Da 1,6-dioxaspiro[4.5]decane-7-butanoic acid, 2-[(2S,2’R,3’S,5R,5’R)-2-ethyloctahydro-3′-methyl-5′-[(2S,3S,5R,6R)-tetrahydro-6-hydroxy-6-(hydroxymethyl)-3,5-dimethyl-2H-pyran-2-yl][2,2′-bifuran]-5-yl]-9-hydroxy-β-methoxy-α,γ,2,8-tetramethyl-, (αS,βR,γS,2S,5R,7S,8R,9S)- 17090-79-8 [RN] 241-154-0 [EINECS] (2S,3R,4S)-4-[(2S,5R,7S,8R,9S)-2-{(2S,2’R,3’S,5R,5’R)-2-Ethyl-5′-[(2S,3S,5R,6R)-6-hydroxy-6-(hydroxymethyl)-3,5-dimethyltetrahydro-2H-pyran-2-yl]-3′-methyloctahydro-2,2′-bifuran-5-yl}-9-hydroxy-2,8-di methyl-1,6-dioxaspiro[4.5]dec-7-yl]-3-methoxy-2-methylpentanoic acid монензин[Russian] مونانسين[Arabic] 莫能星[Chinese] Antibiotic, Antifungal, Antiprotozoal Synonym(s): Monensin A sodium salt Empirical Formula (Hill Notation):C36H61NaO11 CAS Number:22373-78-0 Molecular Weight:692.85 Beilstein:4122200 Title: Monensin CAS Registry Number: 17090-79-8 CAS Name: 2-[5-Ethyltetrahydro-5-[tetrahydro-3-methyl-5-[tetrahydro-6-hydroxy-6-(hydroxymethyl)-3,5-dimethyl-2H-pyran-2-yl]-2-furyl]-2-furyl]-9-hydroxy-b-methoxy-a,g,2,8-tetramethyl-1,6-dioxaspiro[4.5]decane-7-butyric acid Additional Names: monensic acid (obsolete) Manufacturers’ …

SIBUTRAMINE

It’s only fair to share…   SIBUTRAMINE Molecular FormulaC17H26ClN Average mass279.848 Da 1-(4-Chlorophenyl)-N,N-dimethyl-a-(2-methylpropyl)cyclobutane methanamine 1-[1-(4-Chlorophenyl)cyclobutyl]-N,N,3-trimethyl-1-butanamine 106650-56-0 [RN] 106650-56-0 (Sibutramine ); 125494-59-9 (Sibutramine HCl Monohydrate); 84485-00-7 (Sibutramine HCl); 6124 UNII:WV5EC51866, WV5EC51866 сибутрамин[Russian] سيبوترامين[Arabic] 西布曲明[Chinese] Drug Name:Sibutramine Hydrochloride Hydrate Research Code:BTS-54524 Trade Name:Meridia® MOA:Serotonin-norepinephrine reuptake inhibitor Indication:Obesity Status:Withdrawn Company:Abbott (Originator) Sibutramine hydrochloride monohydrate, KES-524, BTS-54524, Meridia, Reductil Sibutramine, formerly …

Difamilast

It’s only fair to share… Difamilast PMDA Moizerto, JAPAN APPROVED 2021/9/27 ジファミラスト ディファミラスト; 地法米司特 N-({2-[4-(difluoromethoxy)-3-(propan-2-yloxy)phenyl]-1,3- oxazol-4-yl}methyl)-2-ethoxybenzamide OPA-15406 Formula C23H24F2N2O5 CAS 937782-05-3 Mol weight 446.4439 MM 36; MM-36-Medimetriks-Pharmaceuticals; Moizerto; OPA-15406 Efficacy Anti-inflammatory, Phosphodiesterase IV inhibitor Comment Treatment of atopic dermatitis OriginatorOtsuka Pharmaceutical Development & Commercialization DeveloperMedimetriks Pharmaceuticals; Otsuka Pharmaceutical Development & Commercialization ClassBenzamides; Nonsteroidal anti-inflammatories; Oxazoles; Skin disorder …

TOLDIMFOS SODIUM

It’s only fair to share…   TOLDIMFOS SODIUM C9H12NNaO2P+  , 220.16 Toldimfos sodium 575-75-7 Sodium (4-(dimethylamino)-2-methylphenyl)phosphinate UNII-6139240O1E sodium;[4-(dimethylamino)-2-methylphenyl]-oxido-oxophosphanium EINECS 209-391-4 C9H13NO2P.Na DTXSID4060361 AKOS015960346 VZ33686 AC-10524 FT-0657398 575-75-7 Sodium (4-(dimethylamino)-2-methylphenyl)phosphinate UNII-6139240O1E sodium;[4-(dimethylamino)-2-methylphenyl]-oxido-oxophosphanium Phosphinic acid, [4-(dimethylamino)-2-methylphenyl]-, sodium salt 6139240O1E Phosphinic acid, (4-(dimethylamino)-2-methylphenyl)-, sodium salt Phosphinic acid, P-(4-(dimethylamino)-2-methylphenyl)-, sodium salt (1:1) Toldimfos is an aromatic phosphorus compound which falls …

Carotegrast methyl

It’s only fair to share… Carotegrast methyl Formula C28H26Cl2N4O5 CAS 401905-67-7 Mol weight 569.4358 PMDA APROVED, CAROGRA, カロテグラストメチル ON 2022/3/28 Antiasthmatic, Integrin alpha 4 inhibitor An alpha4 integrin antagonist. 401905-67-7 [RN] L-Phenylalanine, N-(2,6-dichlorobenzoyl)-4-[6-(dimethylamino)-1,4-dihydro-1-methyl-2,4-dioxo-3(2H)-quinazolinyl]-, methyl ester methyl (2S)-2-[(2,6-dichlorophenyl)formamido]-3-{4-[6-(dimethylamino)-1-methyl-2,4-dioxo-1,2,3,4-tetrahydroquinazolin-3-yl]phenyl}propanoate Methyl N-(2,6-dichlorobenzoyl)-4-[6-(dimethylamino)-1-methyl-2,4-dioxo-1,4-dihydro-3(2H)-quinazolinyl]-L-phenylalaninate Carotegrast Methyl Methyl (2S)-2-(2,6-dichlorobenzamido)-3-{4-[6-(dimethylamino)-1-methyl-2,4-dioxo-1,4-dihydroquinazolin-3(2H)-yl]phenyl}propanoate C28H26Cl2N4O5 : 569.44 [401905-67-7] PATENT WO 2008062859 https://patents.google.com/patent/WO2008062859A1/en       Step 1 (Method 2): The title compound …

Risperidone

It’s only fair to share… Risperidone EU APPROVED 2022/2/14, Okedi   R-64,766 R-64766 RCN-3028 RCN3028 Risperidone, R-64766, Risperdal M-Tab, Risperdal Consta, Rispolept, Belivon, Risperdal Formula C23H27FN4O2 CAS 106266-06-2 Mol weight 410.4845 3-{2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl}-2-methyl-4H,6H,7H,8H,9H-pyrido[1,2-a]pyrimidin-4-one Product Ingredients INGREDIENT UNII CAS INCHI KEY Risperidone tartrate 0S6B72E3LK 666179-92-6 KSWIOGDSXUFKOC-LREBCSMRSA-N Risperidone CAS Registry Number: 106266-06-2 CAS Name: 3-[2-[4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one Manufacturers’ Codes: R-64766 Trademarks: Belivon (Organon); Risperdal (J & …

Lutetium Lu 177 vipivotide tetraxetan

It’s only fair to share… Lutetium Lu 177 vipivotide tetraxetan FDA APPROVED 2022/3/23, Pluvicto To treat prostate-specific membrane antigen-positive metastatic castration-resistant prostate cancer following other therapies Formula C49H65N9O16. Lu. 3H CAS 1703749-62-5 Mol weight 1214.0819 Antineoplastic, Radioactive agent   Disease Prostate cancer (PSMA positive) ルテチウム(177Lu)ビピボチドテトラキセタン; UNII-G6UF363ECX, WHO 11429 G6UF363ECX 177Lu-Psma-617 Vipivotide tetraxetan Lu-177 177Lu-Labeled PSMA-617 2-[4-[2-[[4-[[(2S)-1-[[(5S)-5-carboxy-5-[[(1S)-1,3-dicarboxypropyl]carbamoylamino]pentyl]amino]-3-naphthalen-2-yl-1-oxopropan-2-yl]carbamoyl]cyclohexyl]methylamino]-2-oxoethyl]-7,10-bis(carboxylatomethyl)-1,4,7,10-tetrazacyclododec-1-yl]acetate;lutetium-177(3+) (177Lu)Lutetium 2,2′,2′‘-[10-(2-{[(trans-4-{[(2S)-1-{[(5S)-5-carboxy-5-({[(1S)-1,3-dicarboxypropyl]carbamoyl}amino)pentyl]amino}-3-(2-naphthyl)-1-oxo-2-propanyl]carbamoyl}cyclohexyl)methyl]amino}-2- oxoethyl)-1,4,7,10-tetraazacyclododecane-1,4,7-triyl]triacetate …